Data Sheet

MSDS

CGP77675 [CAS 234772-64-6]

CAS No:	234772-64-6
Applications:	Cancer-Kinase/protease
MW:	443.54
Formula:	C₂₆H₂₉N₅O₂
SMILES:	OC1CCN(CCC2=CC=C(N3C=C(C4=CC=CC(OC)=C4)C5=C(N)N=CN=C53)C=C2)CC1
Purity:	99.00
Description:	CGP77675 is an orally active and potent inhibitor of Src family kinases. CGP77675 inhibits phosphorylation of peptide substrates and autophosphorylation of purified Src (IC50s of 5-20 and 40 nM, respectively), and also inhibits Src, EGFR, KDR, v-Abl, and Lck with IC50s of 5-20, 40, 20, 150, 1000, 310, and 290 nM, respectively. Anticancer activity[1].
Shipping Conditions:	Ship on cold packs
Usage:	Research Use Only