Malantide [CAS 86555-35-3]
Partner: MedChemexpress LLC
CAS No: | 86555-35-3 |
Applications: | Cancer-Kinase/protease |
MW: | 1633.89 |
Formula: | C72H124N22O21 |
SMILES: | O=C(N[C@@H]([C@H](O)C)C(N[C@@H](CCCCN)C(N[C@@H](CCCNC(N)=N)C(N[C@@H](CO)C(NCC(N[C@@H](CO)C(N[C@@H](C(C)C)C(N[C@@H](CC1=CC=C(C=C1)O)C(N[C@@H](CCC(O)=O)C(N2[C@@H](CCC2)C(N[C@@H](CC(C)C)C(N[C@@H](CCCCN)C(N[C@@H]([C@@H](C)CC)C(O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)[C@H](CCCNC(N)=N)N |
Purity: | 98.56 |
Description: | Malantide is a synthetic dodecapeptide derived from the site phosphorylated by cAMP-dependent protein kinase (PKA) on the ?-subunit of phosphorylase kinase. Malantide is a highly specific substrate for PKA with a Km of 15 ?M and shows protein inhibitor (PKI) inhibition >90% substrate phosphorylation in various rat tissue extracts[1]. Malantide is also an efficient substrate for PKC with a Km of 16 ?M[2]. |
Shipping Conditions: | Ship on cold packs |
Usage: | Research Use Only |
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