THZ1 [CAS 1604810-83-4]
Partner: MedChemexpress LLC
| CAS No: | 1604810-83-4 |
| Applications: | Cancer-Kinase/protease |
| MW: | 566.05 |
| Formula: | C31H28ClN7O2 |
| SMILES: | ClC1=CN=C(NC2=CC(NC(C3=CC=C(NC(/C=C/CN(C)C)=O)C=C3)=O)=CC=C2)N=C1C4=CNC5=CC=CC=C54 |
| Purity: | 99.84 |
| Description: | THZ1 is a selective and potent covalent CDK7 inhibitor with an IC50 of 3.2 nM. THZ1 also inhibits the closely related kinases CDK12 and CDK13 and downregulates MYC expression[1][2]. |
| Shipping Conditions: | Ship at ambient |
| Usage: | Research Use Only |
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