PBRM1-BD2-IN-5 [CAS 2819989-61-0]
Partner: MedChemexpress LLC
| CAS No: | 2819989-61-0 |
| MW: | 272.73 |
| Formula: | C15H13ClN2O |
| SMILES: | O=C1NC(C2=CC=CC(C)=C2)NC3=C1C(Cl)=CC=C3 |
| Purity: | 99.55 |
| Description: | PBRM1-BD2-IN-5 is a potent PBRM1 Bromodomain inhibitor with Kd values of 1.5 ?M and 3.9 ?M for PBRM1-BD2 and PBRM1-BD5, respectively, and an IC50 value of 0.26 ?M for PBRM1-BD2. PBRM1-BD2-IN-5 reduces the binding of full-length PBRM1 within the PBAF complex in cell lysates to acetylated histone peptide. PBRM1-BD2-IN-5 can be used to research anticancer[1]. |
| Shipping Conditions: | Ship at ambient |
| Usage: | Research Use Only |
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