1G244 [CAS 847928-32-9]
Partner: MedChemexpress LLC
| CAS No: | 847928-32-9 |
| Applications: | Cancer-Kinase/protease |
| MW: | 504.57 |
| Formula: | C29H30F2N4O2 |
| SMILES: | O=C(N1CC2=C(C=CC=C2)C1)[C@@H](N)CC(N3CCN(C(C4=CC=C(F)C=C4)C5=CC=C(F)C=C5)CC3)=O |
| Purity: | 98.66 |
| Description: | 1G244 is a potent DPP8/9 inhibitor with IC50s of 12 nM and 84 nM, respectively. 1G244 does not inhibit DPPIV and DPPII. 1G244 induces apoptosis in multiple myeloma cells and has anti-myeloma effects[1][2]. |
| Shipping Conditions: | Ship at ambient |
| Usage: | Research Use Only |
Insight Biotechnology Ltd reserves the right to change pricing without notice
