(E/Z)-GSK5182 [CAS 2699724-40-6]
Partner: MedChemexpress LLC
CAS No: | 2699724-40-6 |
MW: | 417.54 |
Formula: | C27H31NO3 |
SMILES: | OCCC/C(C1=CC=CC=C1)=C(C2=CC=C(C=C2)OCCN(C)C)\C3=CC=C(C=C3)O |
Purity: | 99.17 |
Description: | (E/Z)-GSK5182 is a racemic compound of (E)-GSK5182 and (Z)-GSK5182 isomers. GSK5182 is a highly selective and orally active inverse agonist of estrogen-related receptor ? (ERR?) with an IC50 of 79 nM[1]. GSK5182 also induces reactive oxyen species (ROS) generation in hepatocellular carcinoma[1][2][3]. |
Shipping Conditions: | Ship at ambient |
Usage: | Research Use Only |
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