Asimadoline (hydrochloride) [CAS 185951-07-9]
Partner: MedChemexpress LLC
| CAS No: | 185951-07-9 |
| Applications: | Metabolism-protein/nucleotide metabolism |
| MW: | 451.00 |
| Formula: | C27H31ClN2O2 |
| SMILES: | O[C@H]1CCN(C1)C[C@H](C2=CC=CC=C2)N(C)C(C(C3=CC=CC=C3)C4=CC=CC=C4)=O.[H]Cl |
| Purity: | 99.82 |
| Description: | Asimadoline (EMD-61753) hydrochloride is an orally active, selective and peripherally active ?-opioid agonist with IC50s of 5.6 nM (guinea pig) and 1.2 nM (human recombinant). Asimadoline hydrochloride has low permeability across the blood brain barrier and has peripheral anti-inflammatory actions. Asimadoline hydrochloride ameliorates allodynia in diabetic rats and has the potential for irritable bowel syndrome (IBS)[1][2][3]. |
| Shipping Conditions: | Ship at ambient |
| Usage: | Research Use Only |
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