L-365260 [CAS 118101-09-0]
Partner: MedChemexpress LLC
CAS No: | 118101-09-0 |
Applications: | Metabolism-protein/nucleotide metabolism |
MW: | 398.46 |
Formula: | C24H22N4O2 |
SMILES: | O=C(NC1=CC=CC(C)=C1)N[C@H]2C(N(C)C3=CC=CC=C3C(C4=CC=CC=C4)=N2)=O |
Purity: | 99.93 |
Description: | L-365260 is an orally active and selective antagonist of non-peptide gastrin and brain cholecystokinin receptor (CCK-B), with Kis of 1.9 nM and 2.0 nM, respectively. L-365260 interacts in a stereoselective and competitive manner with guinea pig stomach gastrin and brain CCK receptors. L-365260 can enhance Morphine analgesia and prevents Morphine tolerance[1][2][3]. |
Shipping Conditions: | Ship at ambient |
Usage: | Research Use Only |
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