CAY10566 [CAS 944808-88-2]
Partner: MedChemexpress LLC
CAS No: | 944808-88-2 |
Applications: | Cancer-programmed cell death |
MW: | 389.81 |
Formula: | C18H17ClFN5O2 |
SMILES: | CC1=NN=C(C2=NN=C(N3CCC(OC4=CC(F)=CC=C4Cl)CC3)C=C2)O1 |
Purity: | 99.73 |
Description: | CAY10566 is a potent, orally bioavailable and selective stearoyl-CoA desaturase1 (SCD1) inhibitor with IC50s of 4.5 and 26 nM in mouse and human enzymatic assays, respectively.CAY10566 also shows excellent cellular activity in blocking the conversion of saturated long-chain fatty acid-CoAs (LCFA-CoAs) to monounsaturated LCFA-CoAs in HepG2 cells (IC50=7.9 nM or 6.8 nM)[1][2]. |
Shipping Conditions: | Ship at ambient |
Usage: | Research Use Only |
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