Samelisant [CAS 1394808-20-8] (10mM in DMSO)
Partner: MedChemexpress LLC
| CAS No: | 1394808-20-8 |
| Applications: | Neuroscience-Neuromodulation |
| MW: | 446.41 |
| Formula: | C21H33Cl2N3O3 |
| SMILES: | O=C(CN1CCOCC1)NC2=CC=C(C=C2)OC3CCN(CC3)C4CCC4.[H]Cl.[H]Cl |
| Purity: | 98.65 |
| Description: | Samelisant (SUVN-G3031) is a potent and selective histamine H3 receptor (H3R) inverse agonist with good brain penetration and oral bioavailability. Samelisant has a similar binding affinity towards human (hH3R; Ki=8.7 nM) and rat (rH3R;Ki=9.8 nM) H3R indicating no inter-species differences. Samelisant can be used for the research of sleep-related disorders[1]. |
| Shipping Conditions: | Ship on cold packs |
| Usage: | Research Use Only |
Insight Biotechnology Ltd reserves the right to change pricing without notice
