R59949 [CAS 120166-69-0]
Partner: MedChemexpress LLC
| CAS No: | 120166-69-0 |
| Applications: | Cancer-Kinase/protease |
| MW: | 489.58 |
| Formula: | C28H25F2N3OS |
| SMILES: | O=C1N(CCN2CC/C(CC2)=C(C3=CC=C(F)C=C3)\C4=CC=C(F)C=C4)C(NC5=C1C=CC=C5)=S |
| Purity: | 99.08 |
| Description: | R59949 is a pan diacylglycerol kinase (DGK) inhibitor with an IC50 of 300 nM. R59949 strongly inhibits the activity of type I DGK ? and ? and moderately attenuates the activity of type II DGK ? and ?. R59949 activates protein kinase C (PKC) by enhancing the levels of the endogenous ligand diacyl glycerol[1][2][3]. |
| Shipping Conditions: | Ship on cold packs |
| Usage: | Research Use Only |
Insight Biotechnology Ltd reserves the right to change pricing without notice
