Falnidamol [CAS 196612-93-8]
Partner: MedChemexpress LLC
CAS No: | 196612-93-8 |
Applications: | Cancer-Kinase/protease |
MW: | 387.84 |
Formula: | C18H19ClFN7 |
SMILES: | ClC1=CC(NC2=NC=NC3=CN=C(NC(CC4)CCN4C)N=C23)=CC=C1F |
Purity: | 99.05 |
Description: | Falnidamol (BIBX 1382) is an orally active, selective EGFR tyrosine kinase inhibitor with an IC50 of 3 nM. Falnidamol displays > 1000-fold lower potency against ErbB2 (IC50=3.4 ?M) and a range of other related tyrosine kinases (IC50>10 ?M). Falnidamol is a pyrimido-pyrimidine compound and has anti-cancer activity[1][2]. |
Shipping Conditions: | Ship at ambient |
Usage: | Research Use Only |
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